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CHEMISTRYANDPHARMACOLOGY Muraglitazarisanovel,non-thiazolidinedionePPARalpha/gammadualagonist.ItissynthesizedfromoxybenzylglycineandhasshowntohavehighbindingaffinitytothePPARalphaandPPARgammareceptors.Whencomparedwithrosiglitazone,muraglitazarwasfoundtohavecomparablefunctionalactivityatPPARgamma.Whencomparedwithfenofibricacid,aweakPPARalphaagonist,muraglitazarwasfoundtobemorepotentatPPARalpha...[閱讀全文]
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(2005-10-18 13:20:44)
Cholesterol:awaxy,fat-likesubstancepresentineverycellinthebodyandinmanyfoods.Somecholesterolinthebloodisnecessary-butahighlevelcanleadtoheartdisease.[閱讀全文]
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